Strategies for Screening and Characterizing Targeted Covalent Inhibitors

Advancements in drug design have resulted in resurging interest in drugs that form covalent bonds with their targets, often referred to as targeted covalent inhibitors (TCIs). In this webinar, our speakers introduce innovative approaches to screen for covalent binders, including the use of covalent DNA-encoded libraries (DELs), high throughput screening library collections, and covalent fragment libraries for fragment-based hit generation.